Protein Details: P2X purinoceptor 3

Protein ID

ICDB_Pro_0625

Protein Name

P2X purinoceptor 3

Gene Name

P2RX3

Organism

Homo sapiens (Human)

Length

397 amino acids

AlphaFoldDB

AF-P56373-F1-model_v4.pdb

Function

Receptor for ATP that acts as a ligand-gated cation channel. Plays a role in sensory perception. Required for normal perception of pain. Required for normal taste perception (By similarity).

Sequence

MNCISDFFTYETTKSVVVKSWTIGIINRVVQLLIISYFVGWVFLHEKAYQVRDTAIESSVVTKVKGSGLYANRVMDVSDYVTPPQGTSVFVIITKMIVTENQMQGFCPESEEKYRCVSDSQCGPERLPGGGILTGRCVNYSSVLRTCEIQGWCPTEVDTVETPIMMEAENFTIFIKNSIRFPLFNFEKGNLLPNLTARDMKTCRFHPDKDPFCPILRVGDVVKFAGQDFAKLARTGGVLGIKIGWVCDLDKAWDQCIPKYSFTRLDSVSEKSSVSPGYNFRFAKYYKMENGSEYRTLLKAFGIRFDVLVYGNAGKFNIIPTIISSVAAFTSVGVGTVLCDIILLNFLKGADQYKAKKFEEVNETTLKIAALTNPVYPSDQTTAEKQSTDSGAFSIGH

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

BINDING 63..65; /ligand="ATP"; /ligand_id="ChEBI:CHEBI:30616"; /evidence="ECO:0000269|PubMed:27626375;ECO:0007744|PDB:5SVK;ECO:0007744|PDB:5SVL;ECO:0007744|PDB:5SVM;ECO:0007744|PDB:5SVP"; BINDING 172; /ligand="ATP"; /ligand_id="ChEBI:CHEBI:30616"; /evidence="ECO:0000269|PubMed:27626375;ECO:0007744|PDB:5SVK;ECO:0007744|PDB:5SVL;ECO:0007744|PDB:5SVM;ECO:0007744|PDB:5SVP"; BINDING 275; /ligand="ATP"; /ligand_id="ChEBI:CHEBI:30616"; /evidence="ECO:0000269|PubMed:27626375;ECO:0007744|PDB:5SVK;ECO:0007744|PDB:5SVL;ECO:0007744|PDB:5SVM;ECO:0007744|PDB:5SVP"; BINDING 279..281; /ligand="ATP"; /ligand_id="ChEBI:CHEBI:30616"; /evidence="ECO:0000269|PubMed:27626375;ECO:0007744|PDB:5SVK;ECO:0007744|PDB:5SVL;ECO:0007744|PDB:5SVM;ECO:0007744|PDB:5SVP"; BINDING 299; /ligand="ATP"; /ligand_id="ChEBI:CHEBI:30616"; /evidence="ECO:0000269|PubMed:27626375;ECO:0007744|PDB:5SVK;ECO:0007744|PDB:5SVL;ECO:0007744|PDB:5SVM;ECO:0007744|PDB:5SVP"

Disease

Dissociative Amnesia and Chronic Rapidly Progressive Glomerulonephritis

Location

DOI ID

10.1124/mol.51.1.109; 10.1038/nature04632; 10.1101/gr.2596504; 10.1038/nature19367

RefSeq

NP_002550.2; XP_011543371.1; XP_011543372.1

Feature